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AP1189 acetate

CAS No. 959850-74-9

AP1189 acetate( —— )

Catalog No. M28790 CAS No. 959850-74-9

AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    AP1189 acetate
  • Note
    Research use only, not for human use.
  • Brief Description
    AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.
  • Description
    AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.(In Vitro):Added to macrophage cultures, AP1189 reduced cytokine release, an effect reliant on both MC1 and MC3 as evident from the use of Mc1r(-/-) and Mc3r(-/-) macrophages. No melanogenesis was induced by AP1189 in B16-F10 melanocytes.(In Vivo):Oral AP1189 elicited anti-inflammatory actions in peritonitis and, upon administration at the peak of inflammation, accelerated the resolution phase by ～3-fold.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Melanocortin Receptor
  • Recptor
    calmodulin
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    959850-74-9
  • Formula Weight
    358.35
  • Molecular Formula
    C16H18N6O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=[N+](C1=CC=CC=C1N2C(/C=C/C=N/NC(N)=N)=CC=C2)[O-].CC(O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Noriko Koizumi, et al. Combined agent for cell therapy of corneal endothelial cell. US10959997B2
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